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Dictionary learning aims at seeking a dictionary under which the training data can be sparsely represented. Methods in the literature typically formulate the dictionary learning problem as an optimization w.r.t. two variables, i.e.,…

Signal Processing · Electrical Eng. & Systems 2021-10-27 Cheng Cheng , Wei Dai

The emergence of tool-calling-based agent systems introduces a more evidence-driven paradigm for pathology image analysis in contrast to the coarse-grained text-image diagnostic approaches. With the recent large-scale experimental adoption…

Artificial Intelligence · Computer Science 2026-02-24 Haoyang Su , Shaoting Zhang , Xiaosong Wang

LLM agents increasingly operate through multi-turn tool use and environment interaction, where safety risks often emerge from intermediate steps long before they surface in the final outcome. Reactive auditing is therefore insufficient:…

Computation and Language · Computer Science 2026-05-28 Jiaqian Li , Yanshu Li , Boxuan Zhang , Ruixiang Tang , Kuan-Hao Huang

Assessing whether a molecule can be synthesised is a primary task in drug discovery. It enables computational chemists to filter for viable compounds or bias molecular generative models. The notion of synthesisability is dynamic as it…

Biomolecules · Quantitative Biology 2024-04-15 Antonia Calvi , Théophile Gaudin , Dominik Miketa , Dominique Sydow , Liam Wilbraham

Recent advances in autonomous LLM agents demonstrate their ability to improve performance through iterative interaction with the environment. We define this paradigm as Test-Time Improvement (TTI). However, the mechanisms under how and why…

Artificial Intelligence · Computer Science 2026-02-04 Hang Yan , Xinyu Che , Fangzhi Xu , Qiushi Sun , Zichen Ding , Kanzhi Cheng , Jian Zhang , Tao Qin , Jun Liu , Qika Lin

Multi-turn interaction remains challenging for online reinforcement learning. A common solution is trajectory-level optimization, which treats each trajectory as a single training sample. However, this approach can be inefficient and yield…

Artificial Intelligence · Computer Science 2025-11-18 Yuhan Chen , Yuxuan Liu , Long Zhang , Pengzhi Gao , Jian Luan , Wei Liu

We propose Adjustable Molecular Representation (AdaMR), a new large-scale uniform pre-training strategy for small-molecule drugs, as a novel unified pre-training strategy. AdaMR utilizes a granularity-adjustable molecular encoding strategy,…

Biomolecules · Quantitative Biology 2024-04-30 Yan Ding , Hao Cheng , Ziliang Ye , Ruyi Feng , Wei Tian , Peng Xie , Juan Zhang , Zhongze Gu

Large Language Model (LLM) agents are increasingly applied to complex, multi-step tasks that require interaction with diverse external tools across various domains. However, current LLM agent tool planning methods typically rely on greedy,…

Artificial Intelligence · Computer Science 2026-03-16 Shuo Yang , Soyeon Caren Han , Yihao Ding , Shuhe Wang , Eduard Hoy

With the growing imbalance between limited medical resources and escalating demands, AI-based clinical tasks have become paramount. As a sub-domain, medication recommendation aims to amalgamate longitudinal patient history with medical…

Artificial Intelligence · Computer Science 2023-11-28 Xiang Li , Shunpan Liang , Yulei Hou , Tengfei Ma

Two useful strategies to speed up drug development are to increase the patient accrual rate and use novel adaptive designs. Unfortunately, these two strategies often conflict when the evaluation of the outcome cannot keep pace with the…

Methodology · Statistics 2018-07-24 Ruitao Lin , Ying Yuan

Existing works based on molecular knowledge neglect the 3D geometric structure of molecules and fail to learn the high-dimensional information of medications, leading to structural confusion. Additionally, it does not extract key…

Machine Learning · Computer Science 2024-11-13 Shi Mu , Chen Li , Xiang Li , Shunpan Liang

Molecular optimization, aimed at improving binding affinity or other molecular properties, is a crucial task in drug discovery that often relies on the expertise of medicinal chemists. Recently, deep learning-based 3D generative models…

Machine Learning · Computer Science 2025-05-01 Anjie Qiao , Junjie Xie , Weifeng Huang , Hao Zhang , Jiahua Rao , Shuangjia Zheng , Yuedong Yang , Zhen Wang , Guo-Bo Li , Jinping Lei

Optimizing large-language model (LLM) training on distributed domain-specific accelerator systems presents significant challenges due to its complex optimization space. Existing optimization methods, however, rely on time-consuming manual…

Multiagent Systems · Computer Science 2025-11-07 Yuran Ding , Xinwei Chen , Xiaofan Zhang , Zongwei Zhou

This study explores the application and performance of Transformational Machine Learning (TML) in drug discovery. TML, a meta learning algorithm, excels in exploiting common attributes across various domains, thus developing composite…

Biomolecules · Quantitative Biology 2023-10-02 Adnan Mahmud , Oghenejokpeme Orhobor , Ross D. King

The Project Optimus initiative by the FDA's Oncology Center of Excellence is widely viewed as a groundbreaking effort to change the $\textit{status quo}$ of conventional dose-finding strategies in oncology. Unlike in other therapeutic areas…

Applications · Statistics 2023-04-14 Zhenghao Jiang , Gu Mi , Ji Lin , Christelle Lorenzato , Yuan Ji

Emerging reasoning models hold promise for automating scientific discovery. However, their training is hindered by a critical supervision gap: experimental outcomes are abundant, whereas intermediate reasoning steps are rarely documented at…

Biomolecules · Quantitative Biology 2026-03-24 Zequn Liu , Kehan Wu , Shufang Xie , Zekun Guo , Wei Zhang , Tao Qin , Renhe Liu , Yingce Xia

Neural Architecture Search (NAS) has enabled automatic discovery of more efficient neural network architectures, especially for mobile and embedded vision applications. Although recent research has proposed ways of quickly estimating…

Machine Learning · Computer Science 2022-04-28 Saeejith Nair , Saad Abbasi , Alexander Wong , Mohammad Javad Shafiee

LLM-powered agents are emerging as a dominant paradigm for autonomous task solving. Unlike standard inference workloads, agents operate in a strictly serial "LLM-tool" loop, where the LLM must wait for external tool execution at every step.…

Distributed, Parallel, and Cluster Computing · Computer Science 2026-03-20 Yifan Sui , Han Zhao , Rui Ma , Zhiyuan He , Hao Wang , Jianxun Li , Yuqing Yang

Drug discovery is a complex, multi-step pipeline that remains heavily dependent on manual, experience-driven operations; meanwhile, existing customized artificial intelligence tools are fragmented across web applications, desktop software,…

Biomolecules · Quantitative Biology 2026-03-03 Qihua Pan , Dong Xu , Qianwei Yang , Jenna Xinyi Yao , Sisi Yuan , Zexuan Zhu , Jianqiang Li , Junkai Ji

Accurate ADMET (an abbreviation for "absorption, distribution, metabolism, excretion, and toxicity") predictions can efficiently screen out undesirable drug candidates in the early stage of drug discovery. In recent years, multiple…

Biomolecules · Quantitative Biology 2022-05-25 Shanzhuo Zhang , Zhiyuan Yan , Yueyang Huang , Lihang Liu , Donglong He , Wei Wang , Xiaomin Fang , Xiaonan Zhang , Fan Wang , Hua Wu , Haifeng Wang