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Related papers: Binding Free Energies without Alchemy

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This paper applies the Bayesian Model Averaging (BMA) statistical ensemble technique to estimate small molecule solvation free energies. There is a wide range of methods available for predicting solvation free energies, ranging from…

Biomolecules · Quantitative Biology 2016-12-16 Luke J. Gosink , Christopher C. Overall , Sarah M. Reehl , Paul D. Whitney , David L. Mobley , Nathan A. Baker

Flow Matching (FM) models have emerged as a leading paradigm for high-fidelity synthesis. However, their reliance on iterative Ordinary Differential Equation (ODE) solving creates a significant latency bottleneck. Existing solutions face a…

Computer Vision and Pattern Recognition · Computer Science 2026-02-02 Hongxu Chen , Hongxiang Li , Zhen Wang , Long Chen

The scaled boundary finite element method (SBFEM) is a relatively recent boundary element method that allows the approximation of solutions to PDEs without the need of a fundamental solution. A theoretical framework for the convergence…

Numerical Analysis · Mathematics 2021-03-23 Fleurianne Bertrand , Daniele Boffi , Gonzalo G. de Diego

In this work we propose a chemically-informed data-driven approach to benchmark the approximate density-functional tight-binding (DFTB) excited state (ES) methods that are currently available within the DFTB+ suite. By taking advantage of…

Chemical Physics · Physics 2023-01-02 Andrés I. Bertoni , Cristián G. Sánchez

For decades, it was unknown how electron bifurcating systems in Nature prevented energy-wasting short-circuiting reactions that have large driving forces, so synthetic electron bifurcating molecular machines could not be designed and built.…

Biological Physics · Physics 2020-09-09 Jonathon L. Yuly , Peng Zhang , Carolyn E. Lubner , John W. Peters , David N. Beratan

The primary limitation for the application of alchemical free energy methods to a wider variety of complex molecular systems is achieving reasonable sampling. Flexible binding complexes often have high free energy barriers, which require…

Biological Physics · Physics 2026-03-17 Anika Friedman , Michael Shirts

We present a method to explore the free energy landscapes of chemical reactions with post-transition-state bifurcations using an enhanced sampling method based on well-tempered metadynamics. Obviating the need for computationally expensive…

Chemical Physics · Physics 2023-04-18 Juno Nam , YounJoon Jung

The thesis examines in detail the folding and unfolding processes of a number of proteins including hbSBD, DDLNF4, single and multi Ubiquitin. Using simplified coarse-grained off-lattice Go model and CD experiments we have shown the…

Biological Physics · Physics 2013-08-13 Maksim Kouza

Ensemble density functional theory (eDFT) is an exact time-independent alternative to time-dependent DFT (TD-DFT) for the calculation of excitation energies. Despite its formal simplicity and advantages in contrast to TD-DFT (multiple…

Strongly Correlated Electrons · Physics 2017-01-19 Killian Deur , Laurent Mazouin , Emmanuel Fromager

The conformational free energy landscape of a system is a fundamental thermodynamic quantity of importance particularly in the study of soft matter and biological systems, in which the entropic contributions play a dominant role. While…

Biological Physics · Physics 2015-10-13 N. Ramakrishnan , Richard W. Tourdot , Ravi Radhakrishnan

This article fills a gap in the mathematical analysis of Adaptive Biasing algorithms, which are extensively used in molecular dynamics computations. Given a reaction coordinate, ideally, the bias in the overdamped Langevin dynamics would be…

Probability · Mathematics 2019-10-11 Michel Benaïm , Charles-Edouard Bréhier , Pierre Monmarché

This paper studies the distributed optimal bilinear equalizer (OBE) beamforming design for both the uplink and downlink cell-free massive multiple-input multiple-output networks. We consider arbitrary statistics-based channel estimators…

Information Theory · Computer Science 2025-03-04 Zhe Wang , Jiayi Zhang , Hao Lei , Dusit Niyato , Bo Ai

We consider the classical molecular beam epitaxy (MBE) model with logarithmic type potential known as no-slope-selection. We employ a third order backward differentiation (BDF3) in time with implicit treatment of the surface diffusion term.…

Numerical Analysis · Mathematics 2021-10-26 Dong Li , Chaoyu Quan , Wen Yang

Existing works are dedicated to untangling atomized numerical components (features) from the hidden states of Large Language Models (LLMs). However, they typically rely on autoencoders constrained by some training-time regularization on…

Machine Learning · Computer Science 2026-02-13 Hakaze Cho , Haolin Yang , Yanshu Li , Brian M. Kurkoski , Naoya Inoue

We present a novel inference algorithm for arbitrary, binary, undirected graphs. Unlike loopy belief propagation, which iterates fixed point equations, we directly descend on the Bethe free energy. The algorithm consists of two phases,…

Artificial Intelligence · Computer Science 2013-01-14 Max Welling , Yee Whye Teh

This work presents an unfitted boundary algebraic equation (BAE) method for solving three-dimensional elliptic partial differential equations on complex geometries using finite difference on structured meshes. We demonstrate that replacing…

Numerical Analysis · Mathematics 2025-02-11 Qing Xia

Predicting the change in binding free energy ($\Delta \Delta G$) is crucial for understanding and modulating protein-protein interactions, which are critical in drug design. Due to the scarcity of experimental $\Delta \Delta G$ data,…

Computational Engineering, Finance, and Science · Computer Science 2024-10-15 Xiaoran Jiao , Weian Mao , Wengong Jin , Peiyuan Yang , Hao Chen , Chunhua Shen

This work addresses the question of whether it is possible to define simple pair-wise interaction terms to approximate free energies of proteins or polymers. Rather than ask how reliable a potential of mean force is, one can ask how…

Soft Condensed Matter · Physics 2009-10-31 Dirk Reith , Thomas Huber , Florian Mueller-Plathe , Andrew E. Torda

Several research groups have recently reported {\em ab initio} calculations of the melting properties of metals based on density functional theory, but there have been unexpectedly large disagreements between results obtained by different…

Materials Science · Physics 2009-11-07 D. Alfe` , M. J. Gillan , G. D. Price

A thermodynamic integration (TI) protocol incorporating dummy atoms is introduced to calculate free energy differences for disulfide bond formation in proteins. This method successfully reproduces experimental redox potentials for multiple…

Biological Physics · Physics 2025-09-24 Daniel Mejia-Rodriguez , Suman Samantray , Margaret S. Cheung , Hoshin Kim