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AlphaFold has transformed protein structure prediction, but emerging applications such as virtual ligand screening, proteome-wide folding, and de novo binder design demand predictions at a massive scale, where runtime and memory costs…

Because different patients may response quite differently to the same drug or treatment, there is increasing interest in discovering individualized treatment rule. In particular, people are eager to find the optimal individualized treatment…

Methodology · Statistics 2016-04-14 Wei Xiao , Hao Helen Zhang , Wenbin Lu

Generating molecular graphs is crucial in drug design and discovery but remains challenging due to the complex interdependencies between nodes and edges. While diffusion models have demonstrated their potentiality in molecular graph design,…

Machine Learning · Computer Science 2024-11-11 Xiaoyang Hou , Tian Zhu , Milong Ren , Dongbo Bu , Xin Gao , Chunming Zhang , Shiwei Sun

The continuous development of the photovoltaic (PV) industry has raised high requirements for the quality of monocrystalline of PV module cells. When learning to segment defect regions in PV module cell images, Tiny Hidden Cracks (THC) lead…

Computer Vision and Pattern Recognition · Computer Science 2023-10-25 Jianye Yi , Xiaopin Zhong , Weixiang Liu , Zongze Wu , Yuanlong Deng , Zhengguang Wu

Antimicrobial peptides (AMPs) play important roles in cancer, autoimmune diseases, and aging. A critical aspect of AMP functionality is their targeted interaction with pathogen membranes, which often possess altered lipid compositions.…

Multi-cellular robot design aims to create robots comprised of numerous cells that can be efficiently controlled to perform diverse tasks. Previous research has demonstrated the ability to generate robots for various tasks, but these…

Artificial Intelligence · Computer Science 2023-12-04 Heng Dong , Junyu Zhang , Chongjie Zhang

Antigen-antibody binding is a critical process in the immune response. Although recent progress has advanced antibody design, current methods lack a generative framework for end-to-end modeling of full-atom antibody structures and struggle…

Quantitative Methods · Quantitative Biology 2026-02-10 Wenda Wang , Yang Zhang , Zhewei Wei , Wenbing Huang

Protein folding neural networks (PFNNs) such as AlphaFold predict remarkably accurate structures of proteins compared to other approaches. However, the robustness of such networks has heretofore not been explored. This is particularly…

Machine Learning · Computer Science 2023-01-13 Ismail Alkhouri , Sumit Jha , Andre Beckus , George Atia , Alvaro Velasquez , Rickard Ewetz , Arvind Ramanathan , Susmit Jha

Therapeutic antibodies are an essential and rapidly expanding drug modality. The binding specificity between antibodies and antigens is decided by complementarity-determining regions (CDRs) at the tips of these Y-shaped proteins. In this…

Biomolecules · Quantitative Biology 2023-11-29 Fang Wu , Stan Z. Li

We have combined a custom implementation of the fast multiple-time-stepping LN integrator with parallel tempering to explore folding properties of small peptides in implicit solvent on the time scale of microseconds. We applied this…

Biomolecules · Quantitative Biology 2011-08-23 Natha R. Hayre , Rajiv R. P. Singh , Daniel L. Cox

Finite alphabet iterative decoders (FAIDs) for LDPC codes were recently shown to be capable of surpassing the Belief Propagation (BP) decoder in the error floor region on the Binary Symmetric channel (BSC). More recently, the technique of…

Information Theory · Computer Science 2012-07-20 Shiva Kumar Planjery , Bane Vasic , David Declercq

Antimicrobial resistance is one of the biggest health problem, especially in the current period of COVID-19 pandemic. Due to the unique membrane-destruction bactericidal mechanism, antimicrobial peptide-mimetic copolymers are paid more…

Biomolecules · Quantitative Biology 2022-12-09 Tianyu Wu , Yang Tang

It has been reported that the communication cost for synchronizing gradients can be a bottleneck, which limits the scalability of distributed deep learning. Using low-precision gradients is a promising technique for reducing the bandwidth…

Distributed, Parallel, and Cluster Computing · Computer Science 2021-05-18 Ruobing Han , James Demmel , Yang You

Protein binder design is central to therapeutics, diagnostics, and synthetic biology, yet practical deployment remains challenging due to fragmented workflows, high computational costs, and complex tool integration. We present…

Biomolecules · Quantitative Biology 2025-05-29 Jie Gao , Jun Li , Jing Hu , Shanzhuo Zhang , Kunrui Zhu , Yueyang Huang , Xiaonan Zhang , Xiaomin Fang

Target-specific peptides, such as conotoxins, exhibit exceptional binding affinity and selectivity toward ion channels and receptors. However, their therapeutic potential remains underutilized due to the limited diversity of natural…

Biomolecules · Quantitative Biology 2025-05-07 Cheng Ge , Han-Shen Tae , Zhenqiang Zhang , Lu Lu , Zhijie Huang , Yilin Wang , Tao Jiang , Wenqing Cai , Shan Chang , David J. Adams , Rilei Yu

Image edge detection (ED) requires specialized architectures, reliable supervision, and rigorous evaluation criteria to ensure accurate localization. In this work, we present a framework for high-precision ED that jointly addresses…

Computer Vision and Pattern Recognition · Computer Science 2026-02-09 Hao Shu

AI-based protein structure prediction pipelines, such as AlphaFold2, have achieved near-experimental accuracy. These advanced pipelines mainly rely on Multiple Sequence Alignments (MSAs) as inputs to learn the co-evolution information from…

Biomolecules · Quantitative Biology 2023-10-19 Xiaomin Fang , Fan Wang , Lihang Liu , Jingzhou He , Dayong Lin , Yingfei Xiang , Xiaonan Zhang , Hua Wu , Hui Li , Le Song

Generating ligand molecules for specific protein targets, known as structure-based drug design, is a fundamental problem in therapeutics development and biological discovery. Recently, target-aware generative models, especially diffusion…

Biomolecules · Quantitative Biology 2024-10-29 Siyi Gu , Minkai Xu , Alexander Powers , Weili Nie , Tomas Geffner , Karsten Kreis , Jure Leskovec , Arash Vahdat , Stefano Ermon

3D generative models have shown significant promise in structure-based drug design (SBDD), particularly in discovering ligands tailored to specific target binding sites. Existing algorithms often focus primarily on ligand-target binding,…

Structure-based drug design (SBDD), which aims to generate 3D ligand molecules binding to target proteins, is a fundamental task in drug discovery. Existing SBDD methods typically treat protein as rigid and neglect protein structural change…

Biomolecules · Quantitative Biology 2024-10-01 Zaixi Zhang , Mengdi Wang , Qi Liu