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Molecular editing aims to modify a given molecule to optimize desired chemical properties while preserving structural similarity. However, current approaches typically rely on string-based or continuous representations, which fail to…

Machine Learning · Computer Science 2025-05-27 Yuanxin Zhuang , Dazhong Shen , Ying Sun

Recent advances in molecular generative models have demonstrated great promise for accelerating scientific discovery, particularly in drug design. However, these models often struggle to generate high-quality molecules, especially in…

Machine Learning · Computer Science 2025-07-29 Zian Li , Cai Zhou , Xiyuan Wang , Xingang Peng , Muhan Zhang

Federated learning allows distributed medical institutions to collaboratively learn a shared prediction model with privacy protection. While at clinical deployment, the models trained in federated learning can still suffer from performance…

Computer Vision and Pattern Recognition · Computer Science 2021-03-11 Quande Liu , Cheng Chen , Jing Qin , Qi Dou , Pheng-Ann Heng

Structure-based drug design (SBDD) aims to discover drug candidates by finding molecules (ligands) that bind tightly to a disease-related protein (targets), which is the primary approach to computer-aided drug discovery. Recently, applying…

Quantitative Methods · Quantitative Biology 2022-12-01 Tianfan Fu , Wenhao Gao , Connor W. Coley , Jimeng Sun

Diffusion models are a powerful tool for probabilistic forecasting, yet most applications in high-dimensional complex systems predict future states individually. This approach struggles to model complex temporal dependencies and fails to…

Machine Learning · Computer Science 2025-12-10 Salva Rühling Cachay , Miika Aittala , Karsten Kreis , Noah Brenowitz , Arash Vahdat , Morteza Mardani , Rose Yu

Structure-Based molecule optimization (SBMO) aims to optimize molecules with both continuous coordinates and discrete types against protein targets. A promising direction is to exert gradient guidance on generative models given its…

Biomolecules · Quantitative Biology 2025-06-06 Keyue Qiu , Yuxuan Song , Jie Yu , Hongbo Ma , Ziyao Cao , Zhilong Zhang , Yushuai Wu , Mingyue Zheng , Hao Zhou , Wei-Ying Ma

The generation of ligands that both are tailored to a given protein pocket and exhibit a range of desired chemical properties is a major challenge in structure-based drug design. Here, we propose an in-silico approach for the $\textit{de…

Biomolecules · Quantitative Biology 2024-05-27 Julian Cremer , Tuan Le , Frank Noé , Djork-Arné Clevert , Kristof T. Schütt

Generating molecules with high binding affinities to target proteins (a.k.a. structure-based drug design) is a fundamental and challenging task in drug discovery. Recently, deep generative models have achieved remarkable success in…

Biomolecules · Quantitative Biology 2023-05-24 Zaixi Zhang , Qi Liu

Epoxy resins are used extensively in composite materials for a wide range of engineering applications, including structural components of aircraft and spacecraft. The processing of fiber-reinforced epoxy composite structures requires…

Diffusion models have demonstrated strong generative performance; however, generated samples often fail to fully align with human intent. This paper studies a test-time scaling method that enables sampling from regions with higher…

Machine Learning · Computer Science 2026-02-04 Yeongmin Kim , Donghyeok Shin , Byeonghu Na , Minsang Park , Richard Lee Kim , Il-Chul Moon

Electroencephalography (ECoG) offers a promising alternative to conventional electrocorticography (EEG) for the early prediction of Parkinson's disease (PD), providing higher spatial resolution and a broader frequency range. However,…

Machine Learning · Computer Science 2026-02-12 Seongwon Jin , Hanseul Choi , Sunggu Yang , Sungho Park , Jibum Kim

Electroencephalography (EEG)-based multimodal learning integrates brain signals with complementary modalities to improve mental state assessment, providing great clinical potential. The effectiveness of such paradigms largely depends on the…

Machine Learning · Computer Science 2026-05-12 Runhe Zhou , Shanglin Li , Guanxiang Huang , Xinliang Zhou , Qibin Zhao , Motoaki Kawanabe , Yi Ding , Cuntai Guan

A general approach was proposed in this article to develop high-order exponentially fitted basis functions for finite element approximations of multi-dimensional drift-diffusion equations for modeling biomolecular electrodiffusion…

Numerical Analysis · Mathematics 2013-02-13 Melissa R. Swager , Y. C. Zhou

Understanding how small molecules perturb gene expression is essential for uncovering drug mechanisms, predicting off-target effects, and identifying repurposing opportunities. While prior deep learning frameworks have integrated multimodal…

Machine Learning · Computer Science 2026-01-01 Pascal Passigan , Kevin Zhu , Angelina Ning

Structure-based drug design (SBDD) is crucial for developing specific and effective therapeutics against protein targets but remains challenging due to complex protein-ligand interactions and vast chemical space. Although language models…

Biomolecules · Quantitative Biology 2024-08-20 Cong Fu , Xiner Li , Blake Olson , Heng Ji , Shuiwang Ji

Non-reversible Markov chain Monte Carlo schemes based on piecewise deterministic Markov processes have been recently introduced in applied probability, automatic control, physics and statistics. Although these algorithms demonstrate…

Computation · Statistics 2017-08-29 George Deligiannidis , Alexandre Bouchard-Côté , Arnaud Doucet

Machine learning holds tremendous promise for transforming the fundamental practice of scientific discovery by virtue of its data-driven nature. With the ever-increasing stream of research data collection, it would be appealing to…

Machine Learning · Computer Science 2024-03-06 Jianan Fan , Dongnan Liu , Hang Chang , Heng Huang , Mei Chen , Weidong Cai

The ultimate goal of drug design is to find novel compounds with desirable pharmacological properties. Designing molecules retaining particular scaffolds as the core structures of the molecules is one of the efficient ways to obtain…

Quantitative Methods · Quantitative Biology 2019-09-06 Yibo Li , Jianxing Hu , Yanxing Wang , Jielong Zhou , Liangren Zhang , Zhenming Liu

The aim of this paper is to establish exponential mixing of frame flows for convex cocompact hyperbolic manifolds of arbitrary dimension with respect to the Bowen-Margulis-Sullivan measure. Some immediate applications include an asymptotic…

Dynamical Systems · Mathematics 2024-06-28 Pratyush Sarkar , Dale Winter

Molecule generation is advancing rapidly in chemical discovery and drug design. Flow matching methods have recently set the state of the art (SOTA) in unconditional molecule generation, surpassing score-based diffusion models. However,…