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The concept of allostery in which macromolecules switch between two different conformations is a central theme in biological processes ranging from gene regulation to cell signaling to enzymology. Allosteric enzymes pervade metabolic…

Subcellular Processes · Quantitative Biology 2017-01-17 Tal Einav , Linas Mazutis , Rob Phillips

Chemical space exploration underlies drug discovery, yet most generative models treat chemical space as a fixed, implicitly learned distribution, focusing on sampling molecules rather than deliberately designing the space itself. We…

Engineering design optimization seeks to automatically determine the shapes, topologies, or parameters of components that maximize performance under given conditions. This process often depends on physics-based simulations, which are…

Computational Engineering, Finance, and Science · Computer Science 2025-08-12 Florian Felten , Gabriel Apaza , Gerhard Bräunlich , Cashen Diniz , Xuliang Dong , Arthur Drake , Milad Habibi , Nathaniel J. Hoffman , Matthew Keeler , Soheyl Massoudi , Francis G. VanGessel , Mark Fuge

Engineering molecular systems that exhibit complex behavior requires the design of kinetic barriers. For example, an effective catalytic pathway must have a large barrier when the catalyst is absent. While programming such energy barriers…

Emerging Technologies · Computer Science 2020-01-28 Keenan Breik , Cameron Chalk , David Doty , David Haley , David Soloveichik

Modern wearable devices can conveniently record various biosignals in the many different environments of daily living, enabling a rich view of individual health. However, not all biosignals are the same: high-fidelity biosignals, such as…

Machine Learning · Computer Science 2025-02-03 Salar Abbaspourazad , Anshuman Mishra , Joseph Futoma , Andrew C. Miller , Ian Shapiro

Computational prediction of enzyme mechanism and protein function requires accurate physics-based models and suitable sampling. We discuss recent advances in large-scale quantum mechanical (QM) modeling of biochemical systems that have…

Chemical Physics · Physics 2021-05-28 Vyshnavi Vennelakanti , Azadeh Nazemi , Rimsha Mehmood , Adam H. Steeves , Heather J. Kulik

We review enzymatic systems which involve biocatalytic reactions utilized for information processing (biocomputing). Extensive ongoing research in biocomputing, mimicking Boolean logic gates has been motivated by potential applications in…

Biological Physics · Physics 2010-10-12 Evgeny Katz , Vladimir Privman

Protein structure tokenizers (PSTs) are workhorses in protein language modeling, function prediction, and evolutionary analysis. However, existing PSTs only capture local geometry of static structures, and miss the correlated motions and…

Machine Learning · Computer Science 2026-05-15 Kaiwen Shi , Carlos Oliver

Sampling physically valid ligand-binding poses remains a major challenge in molecular docking, particularly for unseen or structurally diverse targets. We introduce PocketVina, a fast and memory-efficient, search-based docking framework…

Quantitative Methods · Quantitative Biology 2025-06-26 Ahmet Sarigun , Bora Uyar , Vedran Franke , Altuna Akalin

Mathematical programming is widely employed across various sectors - such as logistics, energy, and workforce planning - to model and solve industrial optimisation problems, but its use requires substantial domain expertise. Large language…

Programming Languages · Computer Science 2026-05-29 Roberto Rossi , Steven D. Prestwich

Chalcogenide phase-change materials (PCMs) based random access memory (PCRAM) is one of the leading candidates for the development of non-volatile memory and neuro-inspired computing technologies. Recent work shows Indium to be an important…

Materials Science · Physics 2024-06-12 Suyang Sun , Bo Zhang , Xudong Wang , Wei Zhang

Key enzymatic processes in biology use the nonequilibrium error correction mechanism called kinetic proofreading to enhance their specificity. Kinetic proofreading typically requires several dedicated structural features in the enzyme, such…

Molecular Networks · Quantitative Biology 2020-05-26 Vahe Galstyan , Kabir Husain , Fangzhou Xiao , Arvind Murugan , Rob Phillips

Deep learning has transformed protein design, enabling accurate structure prediction, sequence optimization, and de novo protein generation. Advances in single-chain protein structure prediction via AlphaFold2, RoseTTAFold, ESMFold, and…

Machine Learning · Computer Science 2025-02-27 Gregory W. Kyro , Tianyin Qiu , Victor S. Batista

Generative models for molecules based on sequential line notation (e.g. SMILES) or graph representation have attracted an increasing interest in the field of structure-based drug design, but they struggle to capture important 3D spatial…

Machine Learning · Computer Science 2023-12-12 Wei Feng , Lvwei Wang , Zaiyun Lin , Yanhao Zhu , Han Wang , Jianqiang Dong , Rong Bai , Huting Wang , Jielong Zhou , Wei Peng , Bo Huang , Wenbiao Zhou

Proteins are the fundamental macromolecules that play diverse and crucial roles in all living matter and have tremendous implications in healthcare, manufacturing, and biotechnology. Their functions are largely determined by the sequences…

Biomolecules · Quantitative Biology 2024-09-17 Boqiao Lai

In this work, we introduce a polymer discovery platform to efficiently design polymers with tailored properties, exemplified by the discovery of high-performance polymer electrolytes. The platform integrates three core components: a…

Chemical Physics · Physics 2025-04-04 Arash Khajeh , Xiangyun Lei , Weike Ye , Zhenze Yang , Daniel Schweigert , Ha-Kyung Kwon

Configurational entropy is an important factor in the free energy change of many macromolecular recognition and binding processes, and has been intensively studied. Despite great progresses that have been made, the global sampling remains…

Biological Physics · Physics 2012-12-04 Wenzhao Li , Kai Wang , Suyan Tian , Pu Tian

Retrieval-Augmented Generation (RAG) enhances coding tasks by incorporating retrieved code examples into prompts. However, lengthy prompts, often exceeding tens of thousands of tokens, introduce challenges related to limited context windows…

Software Engineering · Computer Science 2026-04-13 Pengfei He , Shaowei Wang , Tse-Hsun Chen

Transformer-based deep learning models are increasingly deployed on energy, and DRAM bandwidth constrained devices such as laptops and gaming consoles, which presents significant challenges in meeting the latency requirements of the models.…

Distributed, Parallel, and Cluster Computing · Computer Science 2025-08-26 Aadesh Deshmukh , Venkata Yaswanth Raparti , Samuel Hsu

The edge partition model (EPM) is a fundamental Bayesian nonparametric model for extracting an overlapping structure from binary matrix. The EPM adopts a gamma process ($\Gamma$P) prior to automatically shrink the number of active atoms.…

Machine Learning · Statistics 2017-09-27 Iku Ohama , Issei Sato , Takuya Kida , Hiroki Arimura