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Related papers: Double-Ended Synthesis Planning with Goal-Constrai…

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Retrosynthetic planning is a critical task in organic chemistry which identifies a series of reactions that can lead to the synthesis of a target product. The vast number of possible chemical transformations makes the size of the search…

Machine Learning · Computer Science 2020-06-30 Binghong Chen , Chengtao Li , Hanjun Dai , Le Song

Retrosynthesis consists of breaking down a chemical compound recursively step-by-step into molecular precursors until a set of commercially available molecules is found with the goal to provide a synthesis route. Its two primary research…

Artificial Intelligence · Computer Science 2024-03-12 Paula Torren-Peraire , Alan Kai Hassen , Samuel Genheden , Jonas Verhoeven , Djork-Arne Clevert , Mike Preuss , Igor Tetko

Goal-directed evaluation of Answer Set Programs is gaining traction thanks to its amenability to create AI systems that can, due to the evaluation mechanism used, generate explanations and justifications. s(CASP) is one of these systems and…

Artificial Intelligence · Computer Science 2021-10-26 Joaquín Arias , Manuel Carro , Gopal Gupta

Retrosynthetic planning is a fundamental task in organic chemistry, yet remains challenging due to its combinatorial complexity. To address this, conventional approaches typically rely on hybrid frameworks that combine single-step…

Artificial Intelligence · Computer Science 2026-04-01 Chenyang Zuo , Siqi Fan , Yizhen Luo , Zaiqing Nie

From medicines to materials, small organic molecules are indispensable for human well-being. To plan their syntheses, chemists employ a problem solving technique called retrosynthesis. In retrosynthesis, target molecules are recursively…

Artificial Intelligence · Computer Science 2018-04-17 Marwin H. S. Segler , Mike Preuss , Mark P. Waller

Asynchronous parallel optimization algorithms for solving large-scale machine learning problems have drawn significant attention from academia to industry recently. This paper proposes a novel algorithm, decoupled asynchronous proximal…

Optimization and Control · Mathematics 2016-05-24 Yitan Li , Linli Xu , Xiaowei Zhong , Qing Ling

Retrosynthesis is the task of breaking down a chemical compound recursively step-by-step into molecular precursors until a set of commercially available molecules is found. Consequently, the goal is to provide a valid synthesis route for a…

Assessing whether a molecule can be synthesised is a primary task in drug discovery. It enables computational chemists to filter for viable compounds or bias molecular generative models. The notion of synthesisability is dynamic as it…

Biomolecules · Quantitative Biology 2024-04-15 Antonia Calvi , Théophile Gaudin , Dominik Miketa , Dominique Sydow , Liam Wilbraham

Constrained bilevel optimization tackles nested structures present in constrained learning tasks like constrained meta-learning, adversarial learning, and distributed bilevel optimization. However, existing bilevel optimization methods…

Optimization and Control · Mathematics 2024-06-05 Wei Yao , Haian Yin , Shangzhi Zeng , Jin Zhang

Dynamic Programming (DP) and Constraint Programming (CP) are well-established paradigms for solving combinatorial optimization problems. Usually, these two approaches are used separately. This paper aims to show that the two can be combined…

Artificial Intelligence · Computer Science 2026-05-25 Emma Legrand , Roger Kameugne , Pierre Schaus

Retrosynthesis, which aims to find a route to synthesize a target molecule from commercially available starting materials, is a critical task in drug discovery and materials design. Recently, the combination of ML-based single-step reaction…

Artificial Intelligence · Computer Science 2024-03-05 Guoqing Liu , Di Xue , Shufang Xie , Yingce Xia , Austin Tripp , Krzysztof Maziarz , Marwin Segler , Tao Qin , Zongzhang Zhang , Tie-Yan Liu

This paper aims to efficiently compute transport maps between probability distributions arising from particle representation of bio-physical problems. We develop a bidirectional DeepParticle (BDP) method to learn and generate solutions…

Computational Physics · Physics 2025-04-17 Tan Zhang , Zhongjian Wang , Jack Xin , Zhiwen Zhang

In container terminal yards, the Container Rehandling Problem (CRP) involves rearranging containers between stacks under specific operational rules, and it is a pivotal optimization challenge in intelligent container scheduling systems.…

Artificial Intelligence · Computer Science 2025-04-22 Ruoqi Wang , Jiawei Li

Designing molecular structures with desired chemical properties is an essential task in drug discovery and material design. However, finding molecules with the optimized desired properties is still a challenging task due to combinatorial…

Biomolecules · Quantitative Biology 2023-02-02 Masatsugu Yamada , Mahito Sugiyama

Automated Synthesis Planning has recently re-emerged as a research area at the intersection of chemistry and machine learning. Despite the appearance of steady progress, we argue that imperfect benchmarks and inconsistent comparisons mask…

Machine Learning · Computer Science 2024-09-09 Krzysztof Maziarz , Austin Tripp , Guoqing Liu , Megan Stanley , Shufang Xie , Piotr Gaiński , Philipp Seidl , Marwin Segler

The classic Resource Constrained Shortest Path (RCSP) problem aims to find a cost optimal path between a pair of nodes in a network such that the resources used in the path are within a given limit. Having been studied for over a decade,…

Artificial Intelligence · Computer Science 2025-04-17 Saman Ahmadi , Andrea Raith , Guido Tack , Mahdi Jalili

Improving the efficiency of Neural Architecture Search (NAS) is a challenging but significant task that has received much attention. Previous works mainly adopted the Differentiable Architecture Search (DARTS) and improved its search…

Computer Vision and Pattern Recognition · Computer Science 2023-12-25 Chongjun Tu , Peng Ye , Weihao Lin , Hancheng Ye , Chong Yu , Tao Chen , Baopu Li , Wanli Ouyang

The canonical solution methodology for finite constrained Markov decision processes (CMDPs), where the objective is to maximize the expected infinite-horizon discounted rewards subject to the expected infinite-horizon discounted costs…

Machine Learning · Computer Science 2020-05-11 Sami Khairy , Prasanna Balaprakash , Lin X. Cai

Past work on optimizing fabrication plans given a carpentry design can provide Pareto-optimal plans trading off between material waste, fabrication time, precision, and other considerations. However, when developing fabrication plans,…

Graphics · Computer Science 2021-08-02 Haisen Zhao , Max Willsey , Amy Zhu , Chandrakana Nandi , Zachary Tatlock , Justin Solomon , Adriana Schulz

Distributed algorithms for solving coupled semidefinite programs (SDPs) commonly require many iterations to converge. They also put high computational demand on the computational agents. In this paper we show that in case the coupled…

Optimization and Control · Mathematics 2015-04-30 Sina Khoshfetrat Pakazad , Anders Hansson , Martin S. Andersen , Anders Rantzer