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A quantum quench is the simplest protocol to investigate nonequilibrium many-body quantum dynamics. Previous studies on the entanglement properties of quenched quantum many-body systems mainly focus on the growth of entanglement entropy.…

Quantum Physics · Physics 2019-07-23 Zongping Gong , Naoto Kura , Masatoshi Sato , Masahito Ueda

Entanglement plays a prominent role in the study of condensed matter many-body systems: Entanglement measures not only quantify the possible use of these systems in quantum information protocols, but also shed light on their physics.…

Quantum Physics · Physics 2021-11-02 Shachar Fraenkel , Moshe Goldstein

Quantum many-body systems realise many different phases of matter characterised by their exotic emergent phenomena. While some simple versions of these properties can occur in systems of free fermions, their occurrence generally implies…

Strongly Correlated Electrons · Physics 2019-10-04 Samuel Spillard , Christopher J. Turner , Konstantinos Meichanetzidis

In this article, we study the kinetics of reversible ligand binding to receptors on a spherical cell surface using a self-consistent stochastic theory. Binding, dissociation, diffusion and rebinding of ligands are incorporated into the…

Subcellular Processes · Quantitative Biology 2009-11-13 Shivam Ghosh , Manoj Gopalakrishnan , Kimberly Forsten-Williams

The binding between proteins and ligands plays a crucial role in the realm of drug discovery. Previous deep learning approaches have shown promising results over traditional computationally intensive methods, but resulting in poor…

Biomolecules · Quantitative Biology 2023-11-29 Shikun Feng , Minghao Li , Yinjun Jia , Weiying Ma , Yanyan Lan

Targeted drug delivery relies on two physical processes: the selective binding of a therapeutic particle to receptors on a specific cell membrane, followed by transport of the particle across the membrane. In this article, we address some…

Soft Condensed Matter · Physics 2021-04-16 Simon Merminod , John R. Edison , Huang Fang , Michael F. Hagan , W. Benjamin Rogers

We extend the Bell forced dissociation rate model to take account into dynamic disorder. The motivation of the present work is from the recent forced dissociation experiments of the adhesive receptor-ligand complexes, in which some…

Soft Condensed Matter · Physics 2007-05-23 Fei Liu , Zhong-can Ou-Yang

Modeling the interaction between proteins and ligands and accurately predicting their binding structures is a critical yet challenging task in drug discovery. Recent advancements in deep learning have shown promise in addressing this…

Machine Learning · Computer Science 2024-01-10 Qizhi Pei , Kaiyuan Gao , Lijun Wu , Jinhua Zhu , Yingce Xia , Shufang Xie , Tao Qin , Kun He , Tie-Yan Liu , Rui Yan

The reduced density matrix of many-body systems possessing an additive conserved quantity can be decomposed in orthogonal sectors which can be independently analyzed. Recently, these have been proven to equally contribute to entanglement…

Statistical Mechanics · Physics 2020-08-05 Xhek Turkeshi , Paola Ruggiero , Vincenzo Alba , Pasquale Calabrese

Cells adapt to changing environments by sensing ligand concentrations using specific receptors. The accuracy of sensing is ultimately limited by the finite number of ligand molecules bound by receptors. Previously derived physical limits to…

Subcellular Processes · Quantitative Biology 2019-11-13 Thierry Mora , Ilya Nemenman

Receptor-ligand binding is a critical first step in signal transduction and the duration of the interaction can impact signal generation. In mammalian cells, clustering of receptors may be facilitated by heterogeneous zones of lipids, known…

Subcellular Processes · Quantitative Biology 2009-11-10 Manoj Gopalakrishnan , Kimberly Forsten-Williams , Matthew A. Nugent , Uwe C. Tauber

We consider a coupled bulk-surface system of partial differential equations with nonlinear coupling modelling receptor-ligand dynamics. The model arises as a simplification of a mathematical model for the reaction between cell surface…

Analysis of PDEs · Mathematics 2016-11-08 Charles M. Elliott , Thomas Ranner , Chandrasekhar Venkataraman

We compute absolute binding affinities for two ligands bound to the FKBP protein using non-equilibrium unbinding simulations. The methodology is straight-forward, requiring little or no modification to many modern molecular simulation…

Biological Physics · Physics 2008-11-24 F. Marty Ytreberg

DNA-encoded library (DEL) screening has revolutionized the detection of protein-ligand interactions through read counts, enabling rapid exploration of vast chemical spaces. However, noise in read counts, stemming from nonspecific…

Machine Learning · Computer Science 2024-12-05 Hanqun Cao , Mutian He , Ning Ma , Chang-yu Hsieh , Chunbin Gu , Pheng-Ann Heng

The adhesion of cells is mediated by receptors and ligands anchored in apposing membranes. A central question is how to characterize the binding affinity of these membrane-anchored molecules. For soluble molecules, the binding affinity is…

Soft Condensed Matter · Physics 2009-06-03 Heinrich Krobath , Bartosz Rozycki , Reinhard Lipowsky , Thomas R. Weikl

We study experimentally accessible lower bounds on entanglement measures based on entropic uncertainty relations. Experimentally quantifying entanglement is highly desired for applications of quantum simulation experiments to fundamental…

Quantum Physics · Physics 2021-05-25 Bjarne Bergh , Martin Gärttner

Accurate prediction of protein-ligand binding affinity is crucial for rapid and efficient drug development. Recently, the importance of predicting binding affinity has led to increased attention on research that models the three-dimensional…

Machine Learning · Computer Science 2024-07-17 Seungyeon Choi , Sangmin Seo , Sanghyun Park

It is widely accepted that the dynamic of entanglement in presence of a generic circuit can be predicted by the knowledge of the statistical properties of the entanglement spectrum. We tested this assumption by applying a Metropolis-like…

Quantum Physics · Physics 2023-09-20 J. Odavić , G. Torre , N. Mijić , D. Davidović , F. Franchini , S. M. Giampaolo

Recent advancements in protein docking site prediction have highlighted the limitations of traditional rigid docking algorithms, like PIPER, which often neglect critical stochastic elements such as solvent-induced fluctuations. These…

Quantitative Methods · Quantitative Biology 2024-12-02 Nanjie Chen , Dongliang Yu , Dmitri Beglov , Mark Kon , Julio Enrique Castrillon-Candas

Many biologically important ligands of proteins are large, flexible, and often charged molecules that bind to extended regions on the protein surface. It is infeasible or expensive to locate such ligands on proteins with standard methods…