English
Related papers

Related papers: Automatic hyperparameter selection in Autodock

200 papers

Virtual screening can accelerate drug discovery by identifying promising candidates for experimental evaluation. Machine learning is a powerful method for screening, as it can learn complex structure-property relationships from experimental…

Machine Learning · Computer Science 2021-02-22 Simon Axelrod , Rafael Gomez-Bombarelli

Predicting the binding structure of a small molecule ligand to a protein -- a task known as molecular docking -- is critical to drug design. Recent deep learning methods that treat docking as a regression problem have decreased runtime…

Biomolecules · Quantitative Biology 2023-02-14 Gabriele Corso , Hannes Stärk , Bowen Jing , Regina Barzilay , Tommi Jaakkola

Accelerating molecular docking -- the process of predicting how molecules bind to protein targets -- could boost small-molecule drug discovery and revolutionize medicine. Unfortunately, current molecular docking tools are too slow to screen…

Optimizing a machine learning pipeline for a task at hand requires careful configuration of various hyperparameters, typically supported by an AutoML system that optimizes the hyperparameters for the given training dataset. Yet, depending…

Machine Learning · Computer Science 2023-10-17 Felix Neutatz , Marius Lindauer , Ziawasch Abedjan

Automatic machine learning (AutoML) is a key enabler of the mass deployment of the next generation of machine learning systems. A key desideratum for future ML systems is the automatic selection of models and hyperparameters. We present a…

Machine Learning · Computer Science 2022-02-22 Moe Kayali , Chi Wang

SkeleDock is a scaffold docking algorithm which uses the structure of a protein-ligand complex as a template to model the binding mode of a chemically similar system. This algorithm was evaluated in the D3R Grand Challenge 4 pose prediction…

Quantitative Methods · Quantitative Biology 2020-05-13 Alejandro Varela-Rial , Maciej Majewski , Alberto Cuzzolin , Gerard Martínez-Rosell , Gianni De Fabritiis

Artificial neural networks have become important to improve the search for admissible string compactifications and characterize them. In this paper we construct the heterotic orbiencoder, a general deep autoencoder to study heterotic…

High Energy Physics - Theory · Physics 2024-01-31 Enrique Escalante-Notario , Ignacio Portillo-Castillo , Saul Ramos-Sanchez

In addition to the best model architecture and hyperparameters, a full AutoML solution requires selecting appropriate hardware automatically. This can be framed as a multi-objective optimization problem: there is not a single best hardware…

Machine Learning · Computer Science 2021-06-11 David Salinas , Valerio Perrone , Olivier Cruchant , Cedric Archambeau

Machine learning algorithms have made remarkable achievements in the field of artificial intelligence. However, most machine learning algorithms are sensitive to the hyper-parameters. Manually optimizing the hyper-parameters is a common…

Machine Learning · Computer Science 2020-03-05 Bozhou Chen , Kaixin Zhang , Longshen Ou , Chenmin Ba , Hongzhi Wang , Chunnan Wang

A stochastic search method, the so-called Adaptive Subspace (AdaSub) method, is proposed for variable selection in high-dimensional linear regression models. The method aims at finding the best model with respect to a certain model…

Computation · Statistics 2021-04-20 Christian Staerk , Maria Kateri , Ioannis Ntzoufras

As a result of the ever increasing complexity of configuring and fine-tuning machine learning models, the field of automated machine learning (AutoML) has emerged over the past decade. However, software implementations like Auto-WEKA and…

Machine Learning · Computer Science 2022-11-09 Dimitrios Iliadis , Marcel Wever , Bernard De Baets , Willem Waegeman

The performance of many algorithms in the fields of hard combinatorial problem solving, machine learning or AI in general depends on tuned hyperparameter configurations. Automated methods have been proposed to alleviate users from the…

Machine Learning · Computer Science 2019-08-23 André Biedenkapp , H. Furkan Bozkurt , Frank Hutter , Marius Lindauer

Retrosynthesis plays a crucial role in the fields of organic synthesis and drug development, where the goal is to identify suitable reactants that can yield a target product molecule. Although existing methods have achieved notable success,…

Machine Learning · Computer Science 2025-10-20 Jiaxi Zhuang , Yu Zhang , Yan Zhang , Ying Qian , Aimin Zhou

Molecular docking, a technique for predicting ligand binding poses, is crucial in structure-based drug design for understanding protein-ligand interactions. Recent advancements in docking methods, particularly those leveraging geometric…

Biomolecules · Quantitative Biology 2024-10-17 Jiaxian Yan , Zaixi Zhang , Jintao Zhu , Kai Zhang , Jianfeng Pei , Qi Liu

A large-scale recommender system usually consists of recall and ranking modules. The goal of ranking modules (aka rankers) is to elaborately discriminate users' preference on item candidates proposed by recall modules. With the success of…

Information Retrieval · Computer Science 2022-05-24 Xinyan Fan , Jianxun Lian , Wayne Xin Zhao , Zheng Liu , Chaozhuo Li , Xing Xie

The performance of modern machine learning methods highly depends on their hyperparameter configurations. One simple way of selecting a configuration is to use default settings, often proposed along with the publication and implementation…

Machine Learning · Statistics 2021-05-03 Florian Pfisterer , Jan N. van Rijn , Philipp Probst , Andreas Müller , Bernd Bischl

Mapping complex metadata structures is crucial in a number of domains such as data integration, ontology alignment or model management. To speed up that process automatic matching systems were developed to compute mapping suggestions that…

Databases · Computer Science 2011-08-10 Eric Peukert , Julian Eberius , Erhard Rahm

We introduce an automatic machine learning (AutoML) modeling architecture called Autostacker, which combines an innovative hierarchical stacking architecture and an Evolutionary Algorithm (EA) to perform efficient parameter search. Neither…

Machine Learning · Computer Science 2018-03-05 Boyuan Chen , Harvey Wu , Warren Mo , Ishanu Chattopadhyay , Hod Lipson

In this paper we investigate an emerging application, 3D scene understanding, likely to be significant in the mobile space in the near future. The goal of this exploration is to reduce execution time while meeting our quality of result…

Computer Vision and Pattern Recognition · Computer Science 2017-03-23 Luigi Nardi , Bruno Bodin , Sajad Saeedi , Emanuele Vespa , Andrew J. Davison , Paul H. J. Kelly

Property Directed Reachability (PDR) is a powerful algorithm for formal verification of hardware and software systems, but its performance is highly sensitive to parameter configurations. Manual parameter tuning is time-consuming and…

Hardware Architecture · Computer Science 2026-04-01 Guangyu Hu , Chen Chen , Xiaofeng Zhou , Jiaxi Zhang , Wei Zhang , Hongce Zhang